SCHEMBL8470595

SCHEMBL8470595

BrC(Br)c1cc2ccccc2c(-c2cccc(I)c2)n1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.35
METAP2 P50579 1/20 0.33
ADORA2A P29274 3/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
PDE4A P27815 2/20 0.32
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8471733 0.85 CYP1A2 (0.36) ABCG2ADORA2AALDH1A1CYP1A2CYP2C9
SCHEMBL10816904 0.84 KDM4E (0.41) ADORA2AALDH1A1
SCHEMBL10983261 0.79 ADORA2A (0.45) ABCG2ADORA2AALDH1A1CYP1A2
SCHEMBL8470699 0.77 ABCG2 (0.37) ABCG2METAP2ADORA2ACHRNB4CHRNA3
SCHEMBL10986562 0.76 KDM4E (0.41) ADORA2AALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8470750 0.76 TSPO (0.45) ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8470649 0.73 ABCG2 (0.35) ABCG2METAP2ADORA2ACHRNB4CHRNA3
SCHEMBL8474142 0.72 PDE4A (0.41) ABCG2ALDH1A1CYP1A2CYP2C19PDE4A
SCHEMBL14018750 0.70 TSPO (0.45) ALDH1A1CYP1A2CYP2C9
SCHEMBL8470642 0.69 PLK1 (0.42) ALDH1A1CYP1A2CYP2C9CYP2C19PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998624-A MEDICAL DIAGNOSIS; BINDING TO SITE OF INJURY, INFLAMMATION EMORY UNIVERSITY (US) 1999-12-07 US disclosed
WO-1998049900-A1 HALOISOQUINOLINE CARBOXAMIDE EMORY UNIVERSITY (US) 1998-11-12 WO disclosed