SCHEMBL8474142

SCHEMBL8474142

O=C(O)c1cc2ccccc2c(-c2cccc(I)c2)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.41
IGFBP3 P17936 1/20 0.40
KDM4E B2RXH2 3/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
GLA P06280 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPK1 P28482 1/20 0.39
MAP2K4 P45985 1/20 0.39
MAPKAPK3 Q16644 1/20 0.39
MAPK6 Q16659 1/20 0.39
ALOX15 P16050 2/20 0.38
TSPO P30536 1/20 0.38
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PDE10A Q9Y233 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10985563 0.86 KDM4E (0.48) IGFBP3KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL8472216 0.85 KDM4E (0.42) IGFBP3KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL8470642 0.84 PLK1 (0.42) PDE4AKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL10995233 0.83 ADORA2A (0.52) IGFBP3MAP2K4PTGER1NR4A1NR4A2
SCHEMBL10986803 0.83 KMO (0.49) PDE4AKDM4EMEN1KMT2AHSD17B10
SCHEMBL10986938 0.80 KMO (0.52) KDM4EMEN1ALDH1A1CYP1A2CYP2C19
SCHEMBL10991830 0.77 LMNA (0.49) KDM4EMEN1ALDH1A1GLAHPGD
SCHEMBL10995427 0.77 DHODH (0.49) KDM4EMEN1KMT2AHSD17B10LMNA
SCHEMBL8470659 0.77 TSPO (0.59) IGFBP3KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL8470699 0.76 ABCG2 (0.37) PDE4AALDH1A1CYP1A2HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998624-A MEDICAL DIAGNOSIS; BINDING TO SITE OF INJURY, INFLAMMATION EMORY UNIVERSITY (US) 1999-12-07 US disclosed
WO-1998049900-A1 HALOISOQUINOLINE CARBOXAMIDE EMORY UNIVERSITY (US) 1998-11-12 WO disclosed