SCHEMBL8470699

SCHEMBL8470699

Cc1cc2ccccc2c(-c2cccc(I)c2)n1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.37
HPGDS O60760 1/20 0.37
CYP1A2 P05177 4/20 0.36
METAP2 P50579 1/20 0.35
ADORA2A P29274 2/20 0.35
CYP2A6 P11509 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NCF1 P14598 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PDE4A P27815 1/20 0.33
LMNA P02545 1/20 0.33
PDE10A Q9Y233 1/20 0.33
CRHR1 P34998 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25847343 0.83 CYP1A2 (0.42) HPGDSCYP1A2ADORA2AALDH1A1HPGD
SCHEMBL8473236 0.83 HPGDS (0.43) HPGDSCYP1A2ADORA2ACYP2A6ALDH1A1
SCHEMBL29118670 0.83 RAB9A (0.43) CYP1A2CYP2A6ALDH1A1HPGDMAPT
SCHEMBL10671008 0.83 PDE10A (0.47) HPGDSCYP1A2ADORA2ACYP2A6ALDH1A1
SCHEMBL29118727 0.81 NPC1 (0.43) ABCG2ALDH1A1HPGDHSD17B10MAPT
SCHEMBL25847342 0.80 HPGDS (0.44) HPGDSCYP1A2ADORA2AALDH1A1HPGD
SCHEMBL17532866 0.79 LMNA (0.46) ABCG2HPGDSCYP1A2HPGDHSD17B10
SCHEMBL29118709 0.78 ALDH1A1 (0.43) HPGDSCYP1A2ADORA2ACYP2A6ALDH1A1
SCHEMBL8470595 0.77 ABCG2 (0.35) ABCG2CYP1A2METAP2ADORA2AALDH1A1
SCHEMBL8470649 0.77 ABCG2 (0.35) ABCG2CYP1A2METAP2ADORA2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117186003-A Preparation method of isoquinoline derivative 苏州大学 2023-12-08 CN disclosed
US-5998624-A MEDICAL DIAGNOSIS; BINDING TO SITE OF INJURY, INFLAMMATION EMORY UNIVERSITY (US) 1999-12-07 US disclosed
WO-1998049900-A1 HALOISOQUINOLINE CARBOXAMIDE EMORY UNIVERSITY (US) 1998-11-12 WO disclosed