SCHEMBL8470734

SCHEMBL8470734

COc1ccc2c(c1F)COCC2=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.45
ALDH1A1 P00352 4/20 0.45
HPGD P15428 2/20 0.45
MAPT P10636 3/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ACHE P22303 3/20 0.39
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
PTPRF P10586 1/20 0.37
CYP2C9 P11712 1/20 0.35
LMNA P02545 2/20 0.33
ADRA1A P35348 1/20 0.33
POLL Q9UGP5 1/20 0.33
HSD17B1 P14061 1/20 0.33
MAPK14 Q16539 1/20 0.33
CYP19A1 P11511 2/20 0.33
TP53 P04637 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28040119 0.82 KDM4E (0.63) KDM4EALDH1A1HPGDMAPTCASP1
SCHEMBL14053635 0.79 KDM4E (0.54) KDM4EALDH1A1HPGDMAPTACHE
SCHEMBL23857698 0.78 KDM4E (0.67) KDM4EALDH1A1HPGDMAPTCASP1
SCHEMBL30815971 0.76 ACHE (0.44) KDM4EALDH1A1HPGDACHEGLA
SCHEMBL22829411 0.76 ACHE (0.44) KDM4EALDH1A1HPGDACHEGLA
SCHEMBL6119284 0.75 ALDH1A1 (0.54) KDM4EALDH1A1HPGDMAPTACHE
SCHEMBL29840331 0.75 ALDH1A1 (0.54) KDM4EALDH1A1HPGDMAPTACHE
SCHEMBL23335828 0.75 ALDH1A1 (0.54) KDM4EALDH1A1HPGDMAPTACHE
SCHEMBL8470376 0.75 KDM4E (0.46) KDM4EALDH1A1HPGDMAPTCASP1
SCHEMBL783942 0.72 ESR1 (0.39) KDM4EALDH1A1HPGDMAPTCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5886016-A ANTIINFLAMMATORY AGENT WITH MINIMAL SIDE EFFECTS FOR TREATING ARTHRITIS G.D. SEARLE & CO. (US) 1999-03-23 US disclosed
US-5670532-A Pyrazolyl derivatives for the treatment of inflammation G. D. SEARLE & CO. (US) 1997-09-23 US disclosed
US-5565482-A ANTIINFLAMMATORY AGENTS, ANTIARTHRITIC AGENTS G.D. SEARLE & CO. (US) 1996-10-15 US disclosed
US-5547975-A ANTIARTHRIC AGENTS, ANALGESICS AND ANTIPYRETICS; INHIBITORS OF CYCLOOXYGENASE II; SIDE EFFECT REDUCTION G.D. SEARLE & CO. 1996-08-20 US disclosed
WO-1996009304-A1 BENZOPYRANOPYRAZOLYL DERIVATIVES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-28 WO disclosed