SCHEMBL8470908

SCHEMBL8470908

COc1cccc(-c2ccc(OC(C)C)cc2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.59
RXRB P28702 1/20 0.59
ABL1 P00519 2/20 0.58
ABCB1 P08183 2/20 0.58
BCR P11274 2/20 0.58
MAOB P27338 2/20 0.53
CYP1A1 P04798 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2E1 P05181 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C8 P10632 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2A6 P11509 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP4B1 P13584 1/20 0.50
CYP2B6 P20813 1/20 0.50
CYP3A5 P20815 1/20 0.50
CYP2A7 P20853 1/20 0.50
CYP3A7 P24462 1/20 0.50
CYP2F1 P24903 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8470898 0.93 RXRA (0.64) RXRARXRBABL1ABCB1BCR
SCHEMBL1180412 0.85 ABL1 (0.77) ABL1ABCB1BCRMAOBCYP1A1
SCHEMBL792197 0.85 ABL1 (0.77) ABL1ABCB1BCRMAOBCYP1A1
SCHEMBL1180343 0.84 ABL1 (0.69) ABL1ABCB1BCRMAOBCYP1A1
SCHEMBL1181204 0.83 ABL1 (0.81) ABL1ABCB1BCRMAOBCYP1A1
SCHEMBL21202067 0.82 ESR2 (0.54) ABL1ABCB1BCRMAOBPTPN5
SCHEMBL8469211 0.81 RXRA (0.72) RXRARXRBMAOBCYP1A2CYP3A4
SCHEMBL9414212 0.81 ABL1 (0.66) ABL1ABCB1BCRMAOBCYP1A1
SCHEMBL13247865 0.81 ABL1 (0.64) ABL1ABCB1BCRMAOBCYP1A1
SCHEMBL178565 0.81 NPSR1 (0.57) RXRARXRBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999025707-A1 2-ARYLBENZO[b]THIOPHENES USEFUL FOR THE TREATMENT OF ESTROGEN DEPRIVATION SYNDROME ELI LILLY AND COMPANY (US) 1999-05-27 WO claimed