SCHEMBL8470898

SCHEMBL8470898

COc1ccc(-c2cccc(OC(C)C)c2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.64
RXRB P28702 1/20 0.64
ABL1 P00519 2/20 0.62
ABCB1 P08183 2/20 0.62
BCR P11274 2/20 0.62
PTPN5 P54829 1/20 0.54
FFAR4 Q5NUL3 3/20 0.51
GABRA1 P14867 1/20 0.50
GABRG2 P18507 1/20 0.50
GABRB3 P28472 1/20 0.50
GABRA5 P31644 1/20 0.50
GABRA3 P34903 1/20 0.50
CYP1A1 P04798 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2E1 P05181 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C8 P10632 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2A6 P11509 1/20 0.50
CYP2C9 P11712 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8470908 0.93 RXRA (0.59) RXRARXRBABL1ABCB1BCR
SCHEMBL8469211 0.85 RXRA (0.72) RXRARXRBPTPN5FFAR4GABRA1
SCHEMBL792197 0.85 ABL1 (0.77) ABL1ABCB1BCRCYP1A1CYP1A2
SCHEMBL1180412 0.85 ABL1 (0.77) ABL1ABCB1BCRCYP1A1CYP1A2
SCHEMBL14303566 0.84 RXRA (0.66) RXRARXRBPTPN5FFAR4GABRA1
SCHEMBL1181204 0.83 ABL1 (0.81) ABL1ABCB1BCRCYP1A1CYP1A2
SCHEMBL21202067 0.82 ESR2 (0.54) ABL1ABCB1BCRPTPN5MAOB
SCHEMBL8524895 0.82 RXRA (0.69) RXRARXRBABL1ABCB1BCR
SCHEMBL14139485 0.81 RXRA (0.59) RXRARXRBPTPN5FFAR4GABRA1
SCHEMBL178565 0.81 NPSR1 (0.57) RXRARXRBCYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999025707-A1 2-ARYLBENZO[b]THIOPHENES USEFUL FOR THE TREATMENT OF ESTROGEN DEPRIVATION SYNDROME ELI LILLY AND COMPANY (US) 1999-05-27 WO claimed
WO-2008087017-A2 NOVEL CASCADE POLYMER COMPLEXES, METHOD FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THE SAME BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-07-24 WO disclosed
WO-1999025707-A1 2-ARYLBENZO[b]THIOPHENES USEFUL FOR THE TREATMENT OF ESTROGEN DEPRIVATION SYNDROME ELI LILLY AND COMPANY (US) 1999-05-27 WO disclosed