SCHEMBL8474378

SCHEMBL8474378

O=C1c2ccccc2C(=O)N1CCN1CCC(c2nsc3cccc(F)c23)CC1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.44
HTR1A P08908 4/20 0.44
HTR2A P28223 4/20 0.44
HTR7 P34969 2/20 0.44
HTR6 P50406 2/20 0.44
DRD3 P35462 1/20 0.42
KDM1A O60341 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1545312 0.80 HTR1D (0.50) DRD2HTR1AHTR2AHTR7HTR6
Hydrochloric Acid SCHEMBL1545002 0.80 HTR1D (0.49) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL8854146 0.79 HTR1A (0.61) DRD2HTR1AHTR2A
SCHEMBL9377355 0.78 HTR1A (0.65) DRD2HTR1AHTR2AHTR7HTR6
Hydrochloric Acid SCHEMBL9381340 0.76 HTR1A (0.62) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL9117307 0.74 HTR1D (0.50) DRD2HTR1AHTR2A
SCHEMBL8787809 0.72 HTR1A (0.41) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL6220554 0.72 HTR1A (0.40) HTR1A
SCHEMBL8858982 0.71 HTR2A (0.57) DRD2HTR1AHTR2AHTR6DRD3
SCHEMBL1545386 0.71 HTR1D (0.47) DRD2HTR1AHTR2AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6001834-A PSYCHOLOGICAL DISORDERS, ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1999-12-14 US disclosed
US-5965546-A ANTIPSYCHOTIC AND ANALGESIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1999-10-12 US disclosed