SCHEMBL8787809

SCHEMBL8787809

O=C1c2ccccc2C(=O)N1CCN1CCC(c2snc3cc(F)ccc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.41
HTR2A P28223 3/20 0.41
DRD2 P14416 2/20 0.41
HTR7 P34969 2/20 0.41
HTR6 P50406 1/20 0.41
KDM1A O60341 1/20 0.40
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8789213 0.94 DRD2 (0.43) HTR1AHTR2ADRD2HTR7HTR6
SCHEMBL1545312 0.82 HTR1D (0.50) HTR1AHTR2ADRD2HTR7HTR6
SCHEMBL9376457 0.81 HTR1A (0.56) HTR1AHTR2ADRD2HTR7HTR6
Hydrochloric Acid SCHEMBL1545002 0.81 HTR1D (0.49) HTR1AHTR2ADRD2HTR7HTR6
SCHEMBL8787429 0.80 DRD2 (0.47) HTR1AHTR2ADRD2ACHE
Hydrochloric Acid SCHEMBL8787530 0.79 DRD2 (0.46) HTR1AHTR2ADRD2ACHE
SCHEMBL8788375 0.76 DRD2 (0.40) HTR2ADRD2HTR7ACHE
SCHEMBL1544931 0.76 ACHE (0.71) HTR1AHTR2ADRD2ACHE
SCHEMBL9117307 0.76 HTR1D (0.50) HTR1AHTR2ADRD2ACHE
SCHEMBL1545242 0.76 HTR1A (0.45) HTR1AHTR2ADRD2HTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP disclosed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP disclosed