SCHEMBL8476129

SCHEMBL8476129

O=C(Nc1c2c(nc3ccccc13)CCCC2)c1ccccc1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.73
GAA P10253 1/20 0.73
KMT2A Q03164 1/20 0.72
MAPT P10636 1/20 0.72
ACHE P22303 5/20 0.67
HDAC6 Q9UBN7 1/20 0.67
HDAC5 Q9UQL6 1/20 0.67
BCHE P06276 4/20 0.60
RIPK1 Q13546 1/20 0.59
KDM4E B2RXH2 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10061487 0.92 HTT (0.67) HTTGAAKMT2AMAPTACHE
SCHEMBL9749208 0.89 HTT (0.64) HTTGAAKMT2AMAPTACHE
SCHEMBL9208663 0.87 HTT (0.74) HTTGAAMAPTACHEBCHE
SCHEMBL8473136 0.86 HTT (0.69) HTTGAAMAPTACHEHDAC6
SCHEMBL8472225 0.85 HTT (0.71) HTTGAAMAPTACHEBCHE
SCHEMBL9747579 0.83 BCHE (0.83) HTTGAAKMT2AMAPTACHE
SCHEMBL8474173 0.83 BCHE (0.66) HTTGAAMAPTACHEBCHE
SCHEMBL9748781 0.82 KDM4E (0.68) HTTGAAKMT2AMAPTACHE
SCHEMBL9382159 0.82 KDM4E (0.65) HTTGAAKMT2AMAPTACHE
SCHEMBL9387187 0.81 KDM4E (0.69) HTTGAAKMT2AMAPTACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861411-A TREATING DISTURBANCES OF MEMORY SUCH AS SENILE DEMENTIA AND ALZHEIMER'S DISEASE MITSUBISHI CHEMICAL CORPORATION (JP) 1999-01-19 US disclosed
US-5536728-A TREATMENT OF SENILE DEMENTIA AND ALZHEIMER'S DISEASE MITSUBISHI CHEMICAL CORPORATION (JP) 1996-07-16 US disclosed
EP-0427636-B1 4-Acylaminopyridine derivatives MITSUBISHI CHEM CORP (JP) 1996-05-29 EP disclosed
US-5397785-A Activators of cholinergic neurons to treat memory disorders such as senile dementia and Alzheimer's disease MITSUBISHI KASEI CORPORATION (JP) 1995-03-14 US disclosed
EP-0319429-B1 9-Acylamino-tetrahydroacridine derivatives and memory enhancing agent containing said derivative as active ingredient MITSUBISHI CHEM IND (JP) 1994-04-27 EP disclosed
US-5175172-A Administering amino-1,2,3,4-tetrahydroacridine and derivatives for elevation of T4 lymphocytes level in patients DIETLIN FRANCOIS (FR) 1992-12-29 US disclosed
EP-0427636-A2 4-Acylaminopyridine derivatives Mitsubishi Chemical Corporation (JP) 1991-05-15 EP disclosed
US-4985430-A ALZHEIMER*S DISEASE MITSUBISHI KASEI CORPORATION (JP) 1991-01-15 US disclosed
EP-0319429-A2 9-Acylamino-tetrahydroacridine derivatives and memory enhancing agent containing said derivative as active ingredient MITSUBISHI KASEI CORPORATION (JP) 1989-06-07 EP disclosed