SCHEMBL8476205

SCHEMBL8476205

N#Cc1ccc(C2(C(=O)O)CC2)cc1F

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APP P05067 9/20 0.52
AKR1C3 P42330 6/20 0.52
AKR1C2 P52895 6/20 0.52
CYP2C19 P33261 6/20 0.52
CYP2C9 P11712 6/20 0.52
CYP3A4 P08684 6/20 0.52
AKR1C1 Q04828 3/20 0.52
CYP2D6 P10635 3/20 0.52
AKR1B10 O60218 1/20 0.50
AKR1C4 P17516 1/20 0.50
PSEN1 P49768 1/20 0.50
PSEN2 P49810 1/20 0.50
APH1B Q8WW43 1/20 0.50
NCSTN Q92542 1/20 0.50
APH1A Q96BI3 1/20 0.50
PSENEN Q9NZ42 1/20 0.50
TRPV4 Q9HBA0 1/20 0.42
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8484905 0.94 APP (0.47) APPAKR1C3AKR1C2CYP2C19CYP2C9
SCHEMBL5886251 0.83 APP (0.40) APPAKR1C3AKR1C2CYP2C19CYP2C9
SCHEMBL5354756 0.82 AR (0.39) APPAKR1C3AKR1C2CYP2C19CYP2C9
SCHEMBL7066508 0.80 APP (0.39) APPAKR1C3AKR1C2CYP2C19CYP2C9
SCHEMBL1465878 0.80 AKR1C3 (0.65) APPAKR1C3AKR1C2CYP2C19CYP2C9
SCHEMBL14446345 0.79 OPRM1 (0.49)
SCHEMBL2198459 0.78 AKR1C3 (0.52) APPAKR1C3AKR1C2CYP2C19CYP2C9
SCHEMBL4823323 0.77 TRPV4 (0.47) TRPV4
SCHEMBL30842826 0.76 APP (0.56) APPAKR1C3AKR1C2CYP2C19CYP2C9
SCHEMBL31759329 0.76 APP (0.69) APPAKR1C3AKR1C2CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1229034-B1 Nicotinamide derivatives and their mimetics as inhibitors of PDE4 isozymes PFIZER PROD INC (US) 2005-04-13 EP disclosed