SCHEMBL8476375

SCHEMBL8476375

O=C(O)C1=Cc2ccccc2C=CS1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 2/20 0.33
DAO P14920 1/20 0.33
TSHR P16473 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
LMNA P02545 1/20 0.31
P4HTM Q9NXG6 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
P2RX4 Q99571 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7520710 0.67 DAO (0.31) NAPRTDAOTSHRALDH1A1ALOX15
Bicarbonate SCHEMBL9350415 0.66 P2RX4 (0.48) NAPRTDAOTSHRALDH1A1ALOX15
SCHEMBL5058579 0.61 GAA (0.35) TSHRLMNA
SCHEMBL29120205 0.60 MAPT (0.45) NAPRTDAOTSHRALDH1A1ALOX15
Phosphine SCHEMBL29120220 0.59
Phenol SCHEMBL28197260 0.59 CA12 (0.69) ALDH1A1ALOX15LMNA
Acrylic Acid SCHEMBL11129651 0.57 LMNA (0.50) NAPRTDAOTSHRALDH1A1ALOX15
SCHEMBL9200523 0.57
SCHEMBL3767165 0.56 MAPT (0.53) TSHRALDH1A1ALOX15MAOAMAOB
SCHEMBL33554 0.56

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1080723-C Production of optically active benzothiepin salts TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-03-13 CN disclosed
US-5952512-A Production of optically active benzothiepin salts TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-09-14 US disclosed
CN-1191538-A Production of optically active benzothiepin salts TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-08-26 CN disclosed
EP-0842179-A1 PRODUCTION OF OPTICALLY ACTIVE BENZOTHIEPIN SALTS Takeda Chemical Industries, Ltd. (JP) 1998-05-20 EP disclosed
WO-1997003989-A1 PRODUCTION OF OPTICALLY ACTIVE BENZOTHIEPIN SALTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-02-06 WO disclosed