SCHEMBL8477162

SCHEMBL8477162

CC(C)(C)[Si](C)(C)OC[C@H](O)CCc1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
FDPS P14324 1/20 0.38
CYP2A6 P11509 1/20 0.38
TBXAS1 P24557 4/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HRH1 P35367 2/20 0.36
ESR1 P03372 1/20 0.36
CYP19A1 P11511 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947288 1.00 CHRNA7 (0.40) CHRNA7L3MBTL1TDP1NPC1RAB9A
SCHEMBL6171825 0.85 DHFR (0.41) MEN1KMT2A
SCHEMBL6171832 0.85 DHFR (0.41) MEN1KMT2A
SCHEMBL6951153 0.82 CHRNA7 (0.43) CHRNA7L3MBTL1TDP1NPC1RAB9A
SCHEMBL8163118 0.78 CHRNA7 (0.39) CHRNA7L3MBTL1TDP1NPC1RAB9A
SCHEMBL7833545 0.78 CHRNA7 (0.39) CHRNA7L3MBTL1TDP1NPC1RAB9A
SCHEMBL6171726 0.78 STAT3 (0.34) NPC1RAB9ACYP2A6
SCHEMBL5016747 0.78 CHRNA7 (0.57) CHRNA7L3MBTL1TDP1CYP2A6TBXAS1
SCHEMBL7978396 0.76 MEN1 (0.36) TDP1NPC1RAB9AKDM4EMEN1
SCHEMBL7978399 0.76 MEN1 (0.36) TDP1NPC1RAB9AKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5977105-A Compounds ASTRA PHARMAEUTICALS LTD. (GB) 1999-11-02 US disclosed
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed