SCHEMBL8478024

SCHEMBL8478024

COc1ccc(C(C(=O)NCl)c2ccc(C(=O)C[N+](=O)[O-])cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
GAA P10253 1/20 0.41
GSK3B P49841 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8480948 0.86 L3MBTL1 (0.42) ALDH1A1L3MBTL1KMT2AMEN1CNR1
SCHEMBL8481390 0.85 CNR1 (0.45) ALDH1A1L3MBTL1KMT2AMEN1CNR1
SCHEMBL8482561 0.84 MEN1 (0.47) ALDH1A1KMT2AMEN1CNR1CNR2
SCHEMBL8478498 0.84 HDAC4 (0.45) L3MBTL1KMT2AMEN1CNR1CNR2
SCHEMBL8482590 0.83 ALDH1A1 (0.37) ALDH1A1L3MBTL1KMT2AMEN1CNR1
SCHEMBL28511885 0.83 ALDH1A1 (0.59) ALDH1A1L3MBTL1KMT2AMEN1GSK3B
SCHEMBL8477772 0.81 HAO1 (0.38) ALDH1A1KMT2AMEN1SMN1; SMN2LMNA
SCHEMBL8479404 0.81 PTPN1 (0.45) CNR2GSK3BHDAC1HDAC8MMP1
SCHEMBL8477689 0.80 MEN1 (0.44) KMT2AMEN1CNR1CNR2HDAC4
SCHEMBL8478094 0.79 ALDH1A1 (0.36) ALDH1A1L3MBTL1KMT2AMEN1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5932765-A REDUCTASE INHIBITORS MERCK PATENT GESELLSCHAFT MIT (DE) 1999-08-03 US disclosed