SCHEMBL8478734

SCHEMBL8478734

COc1ccc(CCCOCC(O)C[N+]2(CC(=O)O)CCNCCN(CC(=O)O)CCN(CC(=O)O)CC2)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.37
ITGB3 P05106 2/20 0.35
ITGA2B P08514 2/20 0.35
DRD2 P14416 1/20 0.35
S1PR1 P21453 1/20 0.34
KCNA3 P22001 1/20 0.34
FKBP1A P62942 3/20 0.33
CHRM5 P08912 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8482377 0.86 L3MBTL1 (0.40) MEN1KMT2A
SCHEMBL8482577 0.83 S1PR1 (0.36) ITGB3ITGA2BS1PR1MEN1KMT2A
SCHEMBL8478303 0.82 ITGB3 (0.39) ITGB3ITGA2BMEN1KMT2A
SCHEMBL8478330 0.81 KDM1A (0.39) MEN1KMT2AALDH1A1
SCHEMBL8541621 0.79 ALDH1A1 (0.50) DRD2MEN1KMT2AALDH1A1
SCHEMBL8478639 0.79 MAPT (0.36) ALDH1A1
SCHEMBL8505430 0.78 SMN1; SMN2 (0.31)
SCHEMBL8478027 0.78 KCNH2 (0.41) KMT2A
SCHEMBL8477737 0.78 MAPT (0.40) ALDH1A1
SCHEMBL8483053 0.78 MAPT (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5871709-A TETRAAZACYCLODODECANE COMPOUNDS SUBSTITUTED WITH ALKYL CARBOXY COMPOUNDS FOR CARDIOVASCULAR DISORDERS AND BRAIN TUMORS SCHERING AKTIENGESELLSCHAFT (DE) 1999-02-16 US disclosed