SCHEMBL8479230

SCHEMBL8479230

NCC(=O)N(c1cccc(F)c1)c1ccccc1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 1/20 0.42
PTPN1 P18031 10/20 0.40
PTGIR P43119 3/20 0.38
PTGER4 P35408 1/20 0.38
PTGER3 P43115 1/20 0.38
PTGER2 P43116 1/20 0.38
PTGDR Q13258 1/20 0.38
DCLRE1B Q9H816 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
LPAR1 Q92633 1/20 0.36
KEAP1 Q14145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8483275 0.85 PTPN1 (0.41) LTB4R2PTPN1
SCHEMBL8485734 0.79 PTPN1 (0.43) PTPN1
SCHEMBL8485704 0.78 PTPN1 (0.42) PTPN1DCLRE1B
SCHEMBL8556010 0.73 RXRA (0.49) PTPN1
SCHEMBL3231875 0.71 NPC1 (0.68) PTPN1
SCHEMBL5696468 0.71 LTB4R2 (0.48) LTB4R2PTPN1
SCHEMBL2094984 0.70 NPSR1 (0.48) PTGIRPTGER4PTGER3PTGER2PTGDR
SCHEMBL10399737 0.70 NPC1 (0.71) PTGIRPTGER4PTGER3PTGER2PTGDR
SCHEMBL1561385 0.69 ALDH1A1 (0.63)
SCHEMBL2094982 0.69 PTGIR (0.47) PTGIRPTGER4PTGER3PTGER2PTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5925647-A TREATMENT OF INSULIN NON-INSULIN DEPENDENT DIABETES SHAMAN PHARMACEUTICALS, INC. (US) 1999-07-20 US disclosed
US-5681958-A TREATMENT OF DIABETES SHAMAN PHARMACEUTICALS, INC. (US) 1997-10-28 US disclosed