SCHEMBL8479802

SCHEMBL8479802

COCCOC(=O)C1=C(C)NC(C)=C(C(=O)OCC2CCCCC2)C1c1cccnc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.59
KDM4E B2RXH2 5/20 0.59
GAA P10253 5/20 0.59
HPGD P15428 5/20 0.59
CASP1 P29466 4/20 0.59
CASP7 P55210 4/20 0.59
HSD17B10 Q99714 4/20 0.59
GLA P06280 1/20 0.59
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
CACNA1B Q00975 1/20 0.52
MAPK1 P28482 2/20 0.50
MAPT P10636 2/20 0.47
ACHE P22303 1/20 0.47
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
LMNA P02545 2/20 0.46
TSHR P16473 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8478622 0.88 ALDH1A1 (0.59) ALDH1A1KDM4EGAAHPGDCASP1
SCHEMBL8478410 0.88 ALDH1A1 (0.59) ALDH1A1KDM4EGAAHPGDCASP1
SCHEMBL8480506 0.87 ALDH1A1 (0.60) ALDH1A1KDM4EGAAHPGDCASP1
SCHEMBL13425331 0.81 MEN1 (0.67) GAAMEN1KMT2ANPSR1
SCHEMBL6952589 0.81 CACNA1C (0.60) GAAMEN1KMT2ACACNA1BMAPT
SCHEMBL6953297 0.79 MEN1 (0.54) GAAMEN1KMT2AMAPTCYP1A2
SCHEMBL7159081 0.78 TSHR (0.70) ALDH1A1KDM4EGAAHPGDCASP1
SCHEMBL7162019 0.78 GAA (0.63) ALDH1A1KDM4EGAAHPGDCASP1
SCHEMBL27386922 0.78 TSHR (0.53) ALDH1A1KDM4EGAAHPGDCASP1
SCHEMBL7161996 0.77 ADORA3 (0.73) ALDH1A1KDM4EGAAHPGDCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6001857-A ADMINISTERING CYCLOPENTYL OR ISOPROPYL 2-METHOXYETHYL 4(2-CHLOROTHIENE-3-YL)-1,4-DIHYDRO-2,6-DIMETHYLPYRIDINE-3,5-DI CARBOXYLATE OR SALT TO TREAT DEPRESSION OR SENILE DEMENTIA IN A PATIENT BAYER AKTIENGESELLSCHAFT (DE) 1999-12-14 US disclosed