SCHEMBL8480253

SCHEMBL8480253

O=S(=O)(c1ccccn1)C1CCNCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.41
CYP3A4 P08684 2/20 0.41
CXCR2 P25025 2/20 0.41
ELOVL6 Q9H5J4 1/20 0.40
ELOVL3 Q9HB03 1/20 0.40
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
NPY5R Q15761 1/20 0.39
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
PLD1 Q13393 1/20 0.38
SLC6A2 P23975 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
LMNA P02545 1/20 0.37
GABRA1 P14867 1/20 0.37
TSHR P16473 1/20 0.37
GABRG2 P18507 1/20 0.37
NFKB1 P19838 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5269173 0.98 HTR6 (0.40) HTR6CYP3A4CXCR2ELOVL6ELOVL3
SCHEMBL28331271 0.88 PKM (0.44) HTR6ELOVL6ELOVL3KDM4EPKM
SCHEMBL13162861 0.78 HTR2A (0.49) HTR6ELOVL6ELOVL3KDM4EPKM
SCHEMBL21652058 0.78 ELOVL6 (0.41) HTR6ELOVL6ELOVL3KDM4EPKM
Piperazine SCHEMBL27620266 0.77 HTR6 (0.44) HTR6CYP3A4KDM4EPKMNPY5R
SCHEMBL24634502 0.77 ELOVL6 (0.46) HTR6ELOVL6ELOVL3KDM4EPKM
SCHEMBL10879779 0.76 ELOVL6 (0.36) HTR6CYP3A4CXCR2ELOVL6ELOVL3
SCHEMBL25391604 0.76 PKM (0.41) ELOVL6ELOVL3KDM4EPKML3MBTL1
SCHEMBL7357127 0.76 PKM (0.41) HTR6CYP3A4ELOVL6ELOVL3KDM4E
SCHEMBL20070379 0.74 NAMPT (0.42) HTR6ELOVL6ELOVL3KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110177786-B Substituted pyrazolo [1,5-A ] pyridine compounds as RET kinase inhibitors 阿雷生物药品公司 2021-12-14 CN disclosed
CN-110177786-A Pyrazolo [1,5-A] pyridine compounds being substituted are as RET kinase inhibitor 阿雷生物药品公司 2019-08-27 CN disclosed
US-5925635-A 2-(OXO-1,3-PERHYDRODIAZEPINES OR 3-OXO-2,3,4,5-TETRAHYDRO-1H-2,4-BENZODIAZEPINES; ANTICOAGULANTS; ENZYME INHIBITORS OF SERINE PROTEASE THROMBIN, KALLIKREIN AND PLASMIN; NERVOUS SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS DUPONT PHARMACEUTICALS COMPANY (US) 1999-07-20 US disclosed