SCHEMBL8480271

SCHEMBL8480271

Fc1ccc2c(c1)[nH]c1c(Cl)c3ccccc3nc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.49
GABRG2 P18507 1/20 0.49
GABRB3 P28472 1/20 0.49
GABRA5 P31644 1/20 0.49
GABRA3 P34903 1/20 0.49
GABRA2 P47869 1/20 0.49
MAPK10 P53779 3/20 0.47
TP53 P04637 3/20 0.47
MAPT P10636 2/20 0.47
MAPK1 P28482 2/20 0.47
NPC1 O15118 2/20 0.47
CASP1 P29466 2/20 0.47
RAB9A P51151 2/20 0.47
CASP7 P55210 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAOA P21397 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8483600 0.89 KDM4E (0.51) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL8483897 0.86 TP53 (0.57) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL8479917 0.84 NPC1 (0.54) GABRA1GABRG2GABRB3GABRA5GABRA3
Hydrochloric Acid SCHEMBL8480319 0.82 NPC1 (0.53) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL8689444 0.78 PTGES (0.49) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL8479326 0.77 GABRP (0.48) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL8483962 0.75 MAOA (0.46) MAPK10NPC1RAB9AMAOAMAOB
SCHEMBL8482652 0.75 PIM1 (0.44) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9232319 0.75 PDE3B (0.48) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL8691082 0.75 KDM4E (0.51) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5925647-A TREATMENT OF INSULIN NON-INSULIN DEPENDENT DIABETES SHAMAN PHARMACEUTICALS, INC. (US) 1999-07-20 US disclosed
US-5681958-A TREATMENT OF DIABETES SHAMAN PHARMACEUTICALS, INC. (US) 1997-10-28 US disclosed