SCHEMBL8481125

SCHEMBL8481125

COC(=O)N1CCC(NC(C)=O)CC1Cc1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.50
CHIT1 Q13231 2/20 0.44
CHIA Q9BZP6 2/20 0.44
CCR5 P51681 1/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
BCL2A1 Q16548 1/20 0.41
TEAD1 P28347 1/20 0.40
OPRK1 P41145 1/20 0.40
LMNA P02545 1/20 0.40
TACR3 P29371 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8481128 1.00 TACR1 (0.50) TACR1CHIT1CHIACCR5MEN1
SCHEMBL7618223 0.88 TACR1 (0.54) TACR1CCR5MEN1KMT2ATEAD1
SCHEMBL7618232 0.88 TACR1 (0.54) TACR1CCR5MEN1KMT2ATEAD1
SCHEMBL7610397 0.83 TACR1 (0.69) TACR1TACR3
SCHEMBL7610403 0.83 TACR1 (0.69) TACR1TACR3
SCHEMBL581154 0.82 CHIT1 (0.43) TACR1CHIT1CHIAOPRK1
SCHEMBL586739 0.82 OPRK1 (0.50) TACR1CHIT1CHIAMEN1KMT2A
SCHEMBL8501936 0.81 TACR1 (0.69) TACR1TACR3
SCHEMBL8501940 0.81 TACR1 (0.69) TACR1TACR3
SCHEMBL8500474 0.81 TACR1 (0.49) TACR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965562-A TREATING DISORDERS INDUCED BY SUBSTANCE P AND MIGRAINE HEADACHE NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
US-5604247-A NEUROKININE ANTAGONIST CIBA-GEIGY CORPORATION (US) 1997-02-18 US disclosed