SCHEMBL8485356

SCHEMBL8485356

O=C1c2ccccc2C(=O)N1CCCOc1ccc(-n2ccnc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.60
RAB9A P51151 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
CYP2D6 P10635 8/20 0.60
CYP2C9 P11712 8/20 0.60
CYP3A4 P08684 7/20 0.60
CYP1A2 P05177 5/20 0.60
CYP2C19 P33261 4/20 0.60
CYP19A1 P11511 1/20 0.60
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA9 Q16790 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487429 0.96 CYP2D6 (0.59) MAPTRAB9ASMN1; SMN2CYP2D6CYP2C9
SCHEMBL8487176 0.95 CYP2D6 (0.57) MAPTRAB9ASMN1; SMN2CYP2D6CYP2C9
SCHEMBL8486062 0.95 CYP2D6 (0.57) MAPTRAB9ASMN1; SMN2CYP2D6CYP2C9
SCHEMBL8619440 0.80 RAB9A (0.77) MAPTRAB9ASMN1; SMN2
SCHEMBL8795375 0.80 CYP2D6 (0.49) CYP2D6CYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL8486023 0.80 CYP2D6 (0.49) CYP2D6CYP2C9CYP3A4CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL8618560 0.79 RAB9A (0.74) MAPTRAB9ASMN1; SMN2
SCHEMBL7299163 0.77 RAB9A (1.00) MAPTRAB9ASMN1; SMN2CYP2D6CYP1A2
SCHEMBL8616243 0.76 RAB9A (0.69) MAPTRAB9ASMN1; SMN2
SCHEMBL9471631 0.76 CYP2D6 (0.77) MAPTCYP2D6CYP2C9CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877196-A N- 4-(imidazolyl or pyrazolyl)phenyl(oxy, sulfinyl, sulfenyl or sulfonyl)alkyl!carboxamides, sulfonamides or phosphoramides having antiarrhythmic properties AMERICAN CYANAMID COMPANY (US) 1999-03-02 US disclosed
EP-0792873-A1 N-(Phenoxyalkyl) carboxamides and their use as antiarrhythmic agents American Cyanamid Company (US) 1997-09-03 EP disclosed