SCHEMBL8795375

SCHEMBL8795375

O=C1c2ccccc2C(=O)N1C/C=C/COc1ccc(-n2ccnc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 9/20 0.49
CYP3A4 P08684 9/20 0.49
CYP2C9 P11712 8/20 0.49
CYP1A2 P05177 5/20 0.49
CYP2C19 P33261 4/20 0.47
CYP19A1 P11511 1/20 0.47
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA9 Q16790 2/20 0.45
PORCN Q9H237 1/20 0.44
MEN1 O00255 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8486023 1.00 CYP2D6 (0.49) CYP2D6CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL8485356 0.80 MAPT (0.60) CYP2D6CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL8487429 0.79 CYP2D6 (0.59) CYP2D6CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL8486062 0.78 CYP2D6 (0.57) CYP2D6CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL8487176 0.78 CYP2D6 (0.57) CYP2D6CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL8794811 0.76 CYP2D6 (0.57) CYP2D6CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL8485506 0.76 CYP2D6 (0.57) CYP2D6CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL9711714 0.75 CYP2D6 (0.61) CYP2D6CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL8486026 0.74 SMN1; SMN2 (0.40) CYP2D6CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL27565923 0.73 TBXAS1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792873-A1 N-(Phenoxyalkyl) carboxamides and their use as antiarrhythmic agents American Cyanamid Company (US) 1997-09-03 EP disclosed