SCHEMBL8485656

SCHEMBL8485656

C=CCc1nnc2c3nc[nH]c3[nH]c(=O)n12

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 2/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8483161 0.75 ADORA2A (0.32) ADORA2BADORA3ADORA2A
SCHEMBL8485775 0.68 NPC1 (0.43)
SCHEMBL8486289 0.64 KDM4E (0.41)
1-Methylxanthine SCHEMBL12037451 0.59 ADORA2A (0.54) ADORA2BADORA3ADORA2A
SCHEMBL9240979 0.59 ADORA2A (0.58) ADORA2BADORA3ADORA2A
Hydrochloric Acid SCHEMBL8345987 0.55 NPSR1 (0.39) ADORA2BADORA3ADORA2A
SCHEMBL8158055 0.54 ADORA2B (0.35) ADORA2BADORA3ADORA2A
SCHEMBL5922505 0.54 ADORA2B (0.35) ADORA2BADORA3ADORA2A
SCHEMBL5134359 0.54 ADORA2A (0.66) ADORA2BADORA3ADORA2A
SCHEMBL4795379 0.53 NPSR1 (0.37) ADORA2BADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990118-A NOVEL PURINE COMPOUNDS AND TRIAZOLOPURINE COMPOUNDS WHICH INHIBIT XANTHINE OXIDASE; REMEDIES FOR HYPERURICEMIA, AND AS PREVENTIVE AND THERAPEUTIC AGENTS FOR GOUT YAMASA CORPORATION (JP) 1999-11-23 US disclosed