SCHEMBL8486996

SCHEMBL8486996

O=S(=O)(c1cc(C(F)(F)F)cc(C(F)(F)F)c1)C1CCNCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.45
ADRB1 P08588 1/20 0.41
CACNA1G O43497 1/20 0.38
CACNA1H O95180 1/20 0.38
PTPN5 P54829 1/20 0.38
CNR1 P21554 1/20 0.37
LMNA P02545 1/20 0.37
CYP3A4 P08684 1/20 0.37
GABRA1 P14867 1/20 0.37
TSHR P16473 1/20 0.37
GABRG2 P18507 1/20 0.37
NFKB1 P19838 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37
GABRA6 Q16445 1/20 0.37
HTR6 P50406 3/20 0.37
TACR1 P25103 4/20 0.36
SLC6A4 P31645 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1498723 0.84 HTR2C (0.54) HTR2CTSHRHTR6
Hydrochloric Acid SCHEMBL1498338 0.83 HTR2C (0.55) HTR2CTSHRHTR6
Hydrochloric Acid SCHEMBL4775615 0.82 HTR2C (0.54) HTR2CHTR6
SCHEMBL16771112 0.75 GABRA1 (0.42) ADRB1CNR1LMNACYP3A4GABRA1
SCHEMBL10207483 0.74 PTGS2 (0.40) CNR1
Hydrochloric Acid SCHEMBL17061868 0.74 GABRA1 (0.41) HTR2CADRB1CNR1LMNACYP3A4
SCHEMBL23061349 0.73 KCNH2 (0.35) CNR1TACR1
SCHEMBL2925179 0.73 STS (0.62) HTR2CCNR1TACR1SLC6A4CES2
SCHEMBL294843 0.72 LMNA (0.39) HTR2CLMNACYP3A4GABRA1TSHR
SCHEMBL25145653 0.71 CACNA1H (0.43) HTR2CCACNA1GCACNA1HTSHRTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5925635-A 2-(OXO-1,3-PERHYDRODIAZEPINES OR 3-OXO-2,3,4,5-TETRAHYDRO-1H-2,4-BENZODIAZEPINES; ANTICOAGULANTS; ENZYME INHIBITORS OF SERINE PROTEASE THROMBIN, KALLIKREIN AND PLASMIN; NERVOUS SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS DUPONT PHARMACEUTICALS COMPANY (US) 1999-07-20 US disclosed