SCHEMBL8487526

SCHEMBL8487526

COC(=O)C1CN(C(=O)OCc2ccccc2)CCN1C(=O)OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.54
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
PDK1 Q15118 1/20 0.53
PDK2 Q15119 1/20 0.53
PDK3 Q15120 1/20 0.53
PDK4 Q16654 1/20 0.53
MMP9 P14780 3/20 0.53
MMP1 P03956 2/20 0.53
MMP3 P08254 2/20 0.53
MMP7 P09237 1/20 0.53
MMP13 P45452 1/20 0.53
HTT P42858 1/20 0.51
PREP P48147 1/20 0.51
NPSR1 Q6W5P4 2/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
CYP2C19 P33261 1/20 0.50
FKBP1A P62942 1/20 0.49
ADAM17 P78536 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20129643 0.91 PARP1 (0.55) SMN1; SMN2NPC1RAB9APDK1PDK2
SCHEMBL13681760 0.91 PARP1 (0.55) SMN1; SMN2NPC1RAB9APDK1PDK2
SCHEMBL6487540 0.91 PDK1 (0.53) SMN1; SMN2NPC1RAB9APDK1PDK2
SCHEMBL1288345 0.91 PDK1 (0.53) SMN1; SMN2NPC1RAB9APDK1PDK2
SCHEMBL15298945 0.91 PDK1 (0.53) SMN1; SMN2NPC1RAB9APDK1PDK2
SCHEMBL2820733 0.91 PARP1 (0.55) SMN1; SMN2NPC1RAB9APDK1PDK2
SCHEMBL19120482 0.89 PDK1 (0.52) SMN1; SMN2NPC1RAB9APDK1PDK2
SCHEMBL15298942 0.89 FKBP1A (0.51) SMN1; SMN2NPC1RAB9APDK1PDK2
SCHEMBL6141635 0.89 FKBP1A (0.51) SMN1; SMN2NPC1RAB9APDK1PDK2
SCHEMBL7802196 0.88 POLB (0.52) SMN1; SMN2NPC1RAB9AHTTPREP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955460-A EFFECTIVE AGAINST INFECTIONS CAUSED BY ANTIBIOTIC RESISTANT BACTERIA PHARMACIA & UPJOHN COMPANY (US) 1999-09-21 US disclosed
US-5922707-A Oxazolidinone antibacterial agent with tricyclic substituents PHARMACIA & UPJOHN COMPANY (US) 1999-07-13 US disclosed