SCHEMBL8488127

SCHEMBL8488127

c1cnc(N2CCN(CCCNc3nccc4ccccc34)CC2)nc1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 4/20 0.64
DRD2 P14416 4/20 0.64
ADRA1A P35348 3/20 0.64
HRH4 Q9H3N8 3/20 0.64
KCNH2 Q12809 1/20 0.64
PDE4B Q07343 2/20 0.51
PDE4D Q08499 2/20 0.51
HTR1A P08908 3/20 0.50
HTR2A P28223 2/20 0.50
ACHE P22303 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8581543 0.96 DRD2 (0.69) DRD3DRD2ADRA1AHRH4KCNH2
Bromide SCHEMBL8484082 0.95 DRD2 (0.68) DRD3DRD2ADRA1AHRH4KCNH2
SCHEMBL8485478 0.93 DRD3 (0.58) DRD3DRD2ADRA1AHRH4KCNH2
SCHEMBL8482786 0.88 DRD2 (0.67) DRD3DRD2ADRA1AHRH4KCNH2
Bromide SCHEMBL8483635 0.87 DRD2 (0.66) DRD3DRD2ADRA1AHRH4KCNH2
Bromide SCHEMBL8485565 0.86 DRD3 (0.62) DRD3DRD2ADRA1AHRH4KCNH2
SCHEMBL8486169 0.82 DRD2 (0.68) DRD3DRD2ADRA1AHRH4KCNH2
SCHEMBL8484819 0.82 DRD2 (0.94) DRD3DRD2ADRA1AHRH4KCNH2
Bromide SCHEMBL8583138 0.81 DRD2 (0.67) DRD3DRD2ADRA1AHRH4KCNH2
SCHEMBL8912854 0.79 HTR1A (0.48) DRD3DRD2ADRA1APDE4BPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999021848-A2 NOVEL 1-(N'-(ARYLALKYLAMINOALKYL))AMINOISOINDOLES; A NEW CLASS OF DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 1999-05-06 WO claimed