SCHEMBL8488159

SCHEMBL8488159

NCCCNS(=O)(=O)c1ccc(N)c2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.59
CYP1A2 P05177 5/20 0.59
CYP2C9 P11712 5/20 0.59
CYP2C19 P33261 5/20 0.59
SCN1A P35498 3/20 0.59
SCN2A Q99250 3/20 0.59
SCN3A Q9NY46 3/20 0.59
ALDH1A1 P00352 2/20 0.59
KDM4E B2RXH2 2/20 0.59
HSD17B10 Q99714 2/20 0.59
NSD2 O96028 6/20 0.58
TP53 P04637 5/20 0.58
CYP2D6 P10635 4/20 0.58
MAPK1 P28482 3/20 0.58
THPO P40225 3/20 0.58
NFKB1 P19838 2/20 0.58
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
PMP22 Q01453 3/20 0.57
NPSR1 Q6W5P4 3/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8968288 0.91 CYP3A4 (0.61) CYP3A4CYP1A2CYP2C9CYP2C19SCN1A
SCHEMBL11573784 0.83 NSD2 (0.59) CYP3A4CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL2013174 0.81 FABP4 (0.71) CYP3A4CYP1A2CYP2C9CYP2C19SCN1A
SCHEMBL11686439 0.81 NSD2 (0.86) CYP3A4CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL9050527 0.79 NSD2 (0.56) CYP2C9CYP2C19NSD2NPSR1TSHR
SCHEMBL3871903 0.78 NSD2 (0.51) CYP3A4CYP1A2CYP2C9CYP2C19SCN1A
SCHEMBL1314962 0.78 NSD2 (0.48) CYP3A4CYP1A2CYP2C9CYP2C19SCN1A
SCHEMBL8488157 0.77 HDAC4 (0.65) CYP3A4CYP1A2CYP2C9CYP2C19SCN1A
SCHEMBL17751328 0.77 NSD2 (0.60) CYP3A4CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL1366996 0.77 NSD2 (0.55) NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999050244-A9 NITROXIDE FREE RADICAL DUAL INDICATOR AGENTS LIPITEK INC (US) 1999-12-09 WO disclosed
WO-1999050244-A1 NITROXIDE FREE RADICAL DUAL INDICATOR AGENTS LIPITEK, INC. (US) 1999-10-07 WO disclosed