SCHEMBL8488477

SCHEMBL8488477

CON(C)C(=O)CCc1cccc2c1OCC2

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.43
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
MTNR1A P48039 6/20 0.38
KDM4C Q9H3R0 1/20 0.37
KCNH2 Q12809 2/20 0.37
CCR8 P51685 1/20 0.37
EED O75530 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
TGM2 P21980 1/20 0.34
KCNA3 P22001 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8488569 0.84 MTNR1A (0.55) MTNR1ASLC6A4
SCHEMBL5521083 0.77 NR3C1 (0.44) PARP1HTR2AHTR2CKDM4C
SCHEMBL12388673 0.75 PARP1 (0.59) PARP1HCRTR1HCRTR2
SCHEMBL28330085 0.73 PARP1 (0.49) PARP1HTR2AHTR2CMTNR1AKDM4C
SCHEMBL17362144 0.73 PARP1 (0.49) PARP1MTNR1AKDM4CKCNH2CCR8
SCHEMBL8489943 0.73 ALDH1A1 (0.36) MTNR1AEEDALDH1A1GAA
SCHEMBL6680529 0.73 PARP1 (0.46) PARP1
SCHEMBL6680532 0.73 PARP1 (0.46) PARP1
SCHEMBL3364106 0.72 PARP1 (0.49) PARP1HTR2AHTR2CMTNR1AKDM4C
SCHEMBL10275022 0.72 PARP1 (0.45) PARP1HTR2AHTR2CMTNR1AKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856529-A ADJUSTMENT OF NERVOUS SYSTEM, ENDOCRINE FUNCTION; REPRODUCTION, BODY WEIGHT AND METABOLISM BRISTOL-MYERS SQUIBB COMPANY (US) 1999-01-05 US disclosed