SCHEMBL8488767

SCHEMBL8488767

Cn1c(OC(=O)c2ccccc2)nc(-c2ccccc2)c1-c1ccncc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
NLRP1 Q9C000 1/20 0.47
RAF1 P04049 1/20 0.44
NSD3 Q9BZ95 1/20 0.44
CNR1 P21554 3/20 0.43
FABP4 P15090 2/20 0.41
FABP5 Q01469 1/20 0.41
MAPK14 Q16539 7/20 0.41
CSNK1D P48730 2/20 0.41
CDC7 O00311 2/20 0.40
DBF4 Q9UBU7 2/20 0.40
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
PTGER1 P34995 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7228732 0.77 RAF1 (0.57) ALDH1A1KDM4EMEN1KMT2ARAF1
SCHEMBL4426390 0.77 RAF1 (0.57) ALDH1A1KDM4EMEN1KMT2ARAF1
SCHEMBL28964533 0.76 BCHE (0.42) ALDH1A1KDM4EMEN1KMT2A
SCHEMBL7445283 0.74 MAPK14 (0.58) FABP4FABP5MAPK14CSNK1DMAPK13
SCHEMBL4422522 0.73 MAPK14 (0.59) MEN1KMT2ANSD3MAPK14CSNK1D
SCHEMBL5079652 0.73 MAPK14 (0.59) MEN1KMT2ANSD3MAPK14CSNK1D
SCHEMBL7415940 0.73 ALDH1A1 (0.56) ALDH1A1KDM4EMEN1KMT2ANSD3
SCHEMBL8488765 0.72 MAPK14 (0.55) ALDH1A1KDM4ENSD3CNR1FABP4
SCHEMBL9961397 0.72 NSD3 (0.55) ALDH1A1KDM4EMEN1KMT2ARAF1
SCHEMBL14369862 0.72 NPC1 (0.55) ALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1083473-A New imidazolium compounds and pharmaceutical composition thereof SMITHKLINE BEECHAM CORP (US) 1994-03-09 CN claimed
US-5916891-A CYTOKINE MEDIATED DISEASES SMITHKLINE BEECHAM CORPORATION (US) 1999-06-29 US disclosed
US-5686455-A Imidazole derivatives and their use as cytokine inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1997-11-11 US disclosed
CN-1083473-A New imidazolium compounds and pharmaceutical composition thereof SMITHKLINE BEECHAM CORP (US) 1994-03-09 CN disclosed