SCHEMBL8489491

SCHEMBL8489491

O=C(O)C1(Br)CC=Cc2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
AKR1C1 Q04828 1/20 0.34
HDAC4 P56524 2/20 0.32
KIF11 P52732 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9155004 0.79 THRB (0.37) THRBTDP1AKR1C1HDAC4KIF11
SCHEMBL461337 0.77 THRB (0.40) THRBTDP1AKR1C1HDAC4KIF11
Hydrochloric Acid SCHEMBL28933194 0.77 THRB (0.36) THRBTDP1AKR1C1HDAC4KIF11
SCHEMBL9899733 0.76 THRB (0.35) THRBTDP1AKR1C1HDAC4KIF11
SCHEMBL8491987 0.76 TDP1 (0.35) THRBTDP1AKR1C1HDAC4KIF11
SCHEMBL9302017 0.76 THRB (0.35) THRBTDP1AKR1C1HDAC4KIF11
SCHEMBL4346969 0.76 THRB (0.35) THRBTDP1AKR1C1HDAC4KIF11
SCHEMBL1126348 0.74 NPC1 (0.32) TDP1
SCHEMBL31186268 0.74 KDM4E (0.34)
SCHEMBL2800949 0.74 KDM4E (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999029670-A2 AMINOCARBONYLTETRALIN AND DIHYDRONAPHTALENE DERIVATES AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-17 WO disclosed
US-5369214-A Method for selective dehalogenation of halogenated polyaromatic compounds THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 1994-11-29 US disclosed