SCHEMBL8489704

SCHEMBL8489704

Cc1nc(N)c2cccc(C)c2c1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.39
CYP1A2 P05177 2/20 0.39
ALDH1A1 P00352 3/20 0.39
LMNA P02545 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.38
HTT P42858 2/20 0.38
RAD52 P43351 2/20 0.38
PSMD14 O00487 1/20 0.38
MITF O75030 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
APEX1 P27695 1/20 0.38
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL509508 0.85 CYP3A4 (0.43) CYP1A2ALDH1A1LMNAKDM4EHPGD
SCHEMBL18497858 0.82 CYP1A2 (0.44) CYP2A6CYP1A2ALDH1A1LMNARAB9A
SCHEMBL12733667 0.76 SMN1; SMN2 (0.50) CYP1A2ALDH1A1LMNARAB9ASMN1; SMN2
SCHEMBL12070710 0.75 KDM4E (0.48) CYP2A6CYP1A2ALDH1A1LMNASMN1; SMN2
SCHEMBL22095249 0.75 LMNA (0.35) CYP2A6CYP1A2ALDH1A1LMNARAB9A
SCHEMBL12490173 0.74 KDM4E (0.42) CYP2A6CYP1A2ALDH1A1LMNARAB9A
SCHEMBL17557169 0.72 LMNA (0.46) CYP2A6CYP1A2ALDH1A1LMNARAB9A
SCHEMBL10434554 0.71 CYP1A2 (0.58) CYP2A6CYP1A2ALDH1A1HPGDMAPT
SCHEMBL27955277 0.71 CYP2A6 (0.46) CYP2A6CYP1A2ALDH1A1LMNARAB9A
SCHEMBL16029928 0.69 CYP2A6 (0.44) CYP2A6CYP1A2ALDH1A1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999011622-A1 AMINO-SUBSTITUTED COMPOUNDS, METHODS, AND COMPOSITIONS FOR INHIBITING PARP ACTIVITY GUILFORD PHARMACEUTICALS INC. (US) 1999-03-11 WO claimed
WO-1999011622-A1 AMINO-SUBSTITUTED COMPOUNDS, METHODS, AND COMPOSITIONS FOR INHIBITING PARP ACTIVITY GUILFORD PHARMACEUTICALS INC. (US) 1999-03-11 WO disclosed