SCHEMBL8490705

SCHEMBL8490705

O=CC=Cc1c[nH]c(C(c2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
ALOX5 P09917 1/20 0.38
MAPK1 P28482 1/20 0.38
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
POLB P06746 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2488026 0.84 P2RX7 (0.32) ALDH1A1KMT2A
SCHEMBL7974226 0.81 KDM4E (0.44) ALDH1A1LMNAMAPK1MEN1NPC1
SCHEMBL8487037 0.78
SCHEMBL7405031 0.75 MAP3K7 (0.44) ALDH1A1LMNAMEN1KMT2A
SCHEMBL7974225 0.73 APP (0.36) LMNAALOX5NPC1
SCHEMBL7978927 0.72 AKR1C3 (0.42)
SCHEMBL12489954 0.71
SCHEMBL7839957 0.69 MAPT (0.48) ALDH1A1LMNAMEN1NPC1KMT2A
SCHEMBL7839951 0.69 HRH3 (0.34) MAPK1
SCHEMBL7375916 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999005114-A2 1H-4(5)-SUBSTITUTED IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS HISTAMINE H3 RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 1999-02-04 WO disclosed