SCHEMBL8494376

SCHEMBL8494376

N#Cc1[nH]nc(-c2cccnc2)c1-c1ccc(N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 2/20 0.51
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
IDO1 P14902 1/20 0.43
LRRK2 Q5S007 1/20 0.43
CYP11B2 P19099 2/20 0.43
RXFP1 Q9HBX9 1/20 0.41
KDM4E B2RXH2 4/20 0.40
MAP2K4 P45985 1/20 0.40
PIM1 P11309 1/20 0.40
ALPL P05186 1/20 0.40
HSD17B10 Q99714 2/20 0.40
HTT P42858 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
MAPT P10636 1/20 0.38
CLK2 P49760 1/20 0.38
CLK3 P49761 1/20 0.38
DYRK1A Q13627 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8491737 0.82 CHRNB2 (0.46) IDO1LRRK2CYP11B2PIM1ALPL
SCHEMBL8490727 0.79 AXL (0.51) AXLADORA2AIDO1LRRK2MAP2K4
SCHEMBL14809869 0.75 ADORA2A (0.58) AXLADORA2AADORA1IDO1LRRK2
SCHEMBL1250789 0.70 CYP11B2 (0.47) ADORA2AADORA1IDO1LRRK2CYP11B2
SCHEMBL16105237 0.70 MAPK14 (0.53) LRRK2
SCHEMBL18745788 0.69 CYP2A6 (0.68) AXLCYP11B2KDM4EHSD17B10HTT
SCHEMBL29818169 0.69 CYP2A6 (0.68) AXLCYP11B2KDM4EHSD17B10HTT
SCHEMBL225149 0.69 CYP2A6 (0.68) AXLCYP11B2KDM4EHSD17B10HTT
SCHEMBL6371302 0.68 AXL (1.00) AXLIDO1LRRK2MAP2K4PIM1
SCHEMBL19943059 0.67 AXL (0.49) AXLIDO1LRRK2CYP11B2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999062885-A1 SUBSTITUTED 1-(4-AMINOPHENYL)PYRAZOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1999-12-09 WO disclosed