SCHEMBL8499685

SCHEMBL8499685

CCCCCC/C=C/c1cccc(Br)c1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.48
CYP2D6 P10635 3/20 0.48
CYP2C19 P33261 3/20 0.48
LMNA P02545 1/20 0.48
POLB P06746 1/20 0.48
CYP2C9 P11712 1/20 0.48
SLC6A19 Q695T7 1/20 0.46
HSD17B3 P37058 1/20 0.44
ALDH1A1 P00352 2/20 0.42
TNNC1 P63316 1/20 0.41
CHRNA7 P36544 1/20 0.40
BACE1 P56817 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10651535 1.00 CYP1A2 (0.48) CYP1A2CYP2D6CYP2C19LMNAPOLB
SCHEMBL8499687 1.00 CYP1A2 (0.48) CYP1A2CYP2D6CYP2C19LMNAPOLB
SCHEMBL10651538 1.00 CYP1A2 (0.48) CYP1A2CYP2D6CYP2C19LMNAPOLB
SCHEMBL8955891 0.93 SLC6A19 (0.48) CYP1A2CYP2D6CYP2C19LMNAPOLB
SCHEMBL8955895 0.93 SLC6A19 (0.48) CYP1A2CYP2D6CYP2C19LMNAPOLB
SCHEMBL9305792 0.85 CYP1A2 (0.55) CYP1A2CYP2D6CYP2C19LMNAPOLB
SCHEMBL10742837 0.81 LCK (0.49) TNNC1
SCHEMBL10753147 0.81 LCK (0.49) TNNC1
SCHEMBL16974816 0.81 LCK (0.49) TNNC1
SCHEMBL16679898 0.81 LCK (0.49) TNNC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108017592-A A kind of synthetic method of cis-1,1- cyclopropane dicarboxylic acids diethylester 亳州学院 2018-05-11 CN disclosed
US-5952316-A FOR TREATING AUTOIMMUNE DISEASES, E.G., RHEUMATIOD ARTHRITIS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1999-09-14 US disclosed
EP-0627406-B1 2-AMINO-1,3-PROPANEDIOL COMPOUND AND IMMUNOSUPPRESSANT YOSHITOMI PHARMACEUTICAL (JP) 1998-10-28 EP disclosed
US-5719176-A 2-amino-1,3-propanediol compound and immunosuppressant YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1998-02-17 US disclosed
US-5604229-A 2-amino-1,3-propanediol compound and immunosuppressant YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-02-18 US disclosed
EP-0627406-A1 2-AMINO-1,3-PROPANEDIOL COMPOUND AND IMMUNOSUPPRESSANT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-12-07 EP disclosed