SCHEMBL8499951

SCHEMBL8499951

C=C(C(=O)OC)c1c(C)ncn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.36
MEN1 O00255 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
KMT2A Q03164 1/20 0.32
SIRT2 Q8IXJ6 6/20 0.31
KDM4E B2RXH2 1/20 0.31
CES1 P23141 1/20 0.31
HPGD P15428 2/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
TSHR P16473 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
HIF1A Q16665 1/20 0.30
HSD17B10 Q99714 1/20 0.30
CASP3 P42574 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2236527 0.73 KDM4E (0.40) KCNN4MEN1KMT2AKDM4ELMNA
SCHEMBL8499551 0.73 SIRT2 (0.42) KCNN4SIRT2
SCHEMBL8499957 0.71 L3MBTL1 (0.40) KCNN4MEN1KMT2AKDM4ELMNA
SCHEMBL7412278 0.71 L3MBTL1 (0.40) KCNN4MEN1KMT2AKDM4ELMNA
SCHEMBL2233946 0.70 KCNN4 (0.36) KCNN4MEN1KMT2AKDM4ETSHR
SCHEMBL1424040 0.70 CDC25B (0.47) MEN1KMT2AKDM4EHPGDTSHR
SCHEMBL10439557 0.70 CYP11B1 (0.37) KCNN4MEN1OPRM1OPRD1KMT2A
SCHEMBL10439558 0.69 CYP1A2 (0.44) KCNN4MEN1OPRM1OPRD1KMT2A
SCHEMBL7534704 0.69 HIF1A (0.37) MEN1KMT2AKDM4EHPGDALDH1A1
SCHEMBL9756933 0.67 MEN1 (0.37) KCNN4MEN1KMT2ASIRT2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5932606-A Pyrazinone, pyridinone, piperidine and pyrrolidine thrombin inhibitors MERCK & CO., INC. (US) 1999-08-03 US disclosed