SCHEMBL8500385

SCHEMBL8500385

CCC(=O)Oc1ccc(Oc2c(-c3cccc(OC)c3)ccc3ccccc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
MTNR1A P48039 6/20 0.43
MTNR1B P49286 5/20 0.43
GPR84 Q9NQS5 1/20 0.42
DGAT2 Q96PD7 3/20 0.42
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP1B1 Q16678 1/20 0.40
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
HTR2C P28335 2/20 0.40
MCL1 Q07820 1/20 0.40
BAD Q92934 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
BRD4 O60885 1/20 0.40
CNR2 P34972 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8502205 0.93 MTNR1A (0.43) TDP1L3MBTL1MTNR1AMTNR1BGPR84
SCHEMBL8497554 0.89 L3MBTL1 (0.51) TDP1L3MBTL1GPR84TP53MAPT
SCHEMBL8500568 0.89 ESR1 (0.48) MTNR1AMTNR1BTHRATHRB
SCHEMBL8500292 0.88 ESR1 (0.47) TDP1L3MBTL1THRATHRBTP53
SCHEMBL8501340 0.88 ELANE (0.48) TDP1L3MBTL1TP53MAPTELANE
SCHEMBL8497702 0.85 ESR1 (0.49) MTNR1AMTNR1BCYP1A2THRATHRB
SCHEMBL8497439 0.85 ESR1 (0.49) MTNR1AMTNR1BDGAT2AKR1C3AKR1C2
SCHEMBL6050235 0.83 MIF (0.46) GPR84CYP1A1CYP1A2CYP1B1BRD4
SCHEMBL8500300 0.82 CYP1A2 (0.40) TDP1L3MBTL1MTNR1AMTNR1BGPR84
SCHEMBL8501206 0.82 MAPT (0.45) TDP1L3MBTL1TP53MAPTELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed