SCHEMBL8501020

SCHEMBL8501020

Cc1cccnc1-n1ccnc1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.53
CYP2E1 P05181 1/20 0.53
CYP2A6 P11509 1/20 0.53
ALDH1A1 P00352 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP19A1 P11511 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAPK1 P28482 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HSD11B1 P28845 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27536382 0.81 CYP3A4 (0.39) CYP3A4CYP2E1CYP2A6ALDH1A1NPSR1
SCHEMBL8498623 0.81 CYP3A4 (0.50) CYP3A4CYP2E1CYP2A6ALDH1A1CYP1A2
SCHEMBL8498987 0.81 RPS6KA5 (0.39) CYP3A4CYP2E1CYP2A6NPSR1NOS3
SCHEMBL8089304 0.81 CYP3A4 (0.39) CYP3A4CYP2E1CYP2A6ALDH1A1NPSR1
SCHEMBL8502061 0.79 CYP3A4 (0.47) CYP3A4CYP2E1CYP2A6ALDH1A1CYP1A2
SCHEMBL8733365 0.79 CYP3A4 (0.47) CYP3A4CYP2E1CYP2A6ALDH1A1CYP1A2
SCHEMBL7130873 0.78 CYP2E1 (0.46) CYP3A4CYP2E1CYP2A6ALDH1A1KDM4E
SCHEMBL12926022 0.76 CYP3A4 (0.52) CYP3A4CYP2E1CYP2A6ALDH1A1CYP1A2
SCHEMBL19080612 0.75 CYP3A4 (0.44) CYP3A4CYP2E1CYP2A6ALDH1A1CYP1A2
SCHEMBL14428964 0.74 CYP3A4 (0.50) CYP3A4CYP2E1CYP2A6ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946559-A2 IMIDAZOPYRIDAZINES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1999-10-06 EP disclosed
WO-1998028299-A2 IMIDAZOPYRIDAZINES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-07-02 WO disclosed