SCHEMBL8498623

SCHEMBL8498623

Cc1nccn1-c1ncccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.50
CYP2E1 P05181 1/20 0.50
CYP2A6 P11509 1/20 0.50
TRPV1 Q8NER1 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD11B1 P28845 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ICMT O60725 1/20 0.38
GRM5 P41594 1/20 0.38
RPS6KA5 O75582 2/20 0.38
CYP17A1 P05093 1/20 0.36
KDR P35968 1/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8501020 0.81 CYP3A4 (0.53) CYP3A4CYP2E1CYP2A6CYP1A2CYP2D6
SCHEMBL8500406 0.81 RPS6KA5 (0.40) TRPV1HSD11B1RPS6KA5
SCHEMBL12528529 0.79 TRPV1 (0.41) TRPV1CYP1A2HSD11B1RPS6KA5CYP17A1
SCHEMBL8498621 0.79 RPS6KA5 (0.38) TRPV1HSD11B1RPS6KA5
SCHEMBL12342913 0.76 CYP3A4 (0.47) CYP3A4CYP2E1CYP2A6CYP1A2CYP2D6
SCHEMBL8502061 0.76 CYP3A4 (0.47) CYP3A4CYP2E1CYP2A6CYP1A2CYP2D6
SCHEMBL8733365 0.76 CYP3A4 (0.47) CYP3A4CYP2E1CYP2A6CYP1A2CYP2D6
SCHEMBL7130873 0.75 CYP2E1 (0.46) CYP3A4CYP2E1CYP2A6HSD11B1ALDH1A1
SCHEMBL10757865 0.73 CYP2E1 (0.38) CYP3A4CYP2E1CYP2A6TRPV1ALDH1A1
SCHEMBL12528652 0.72 TRPV1 (0.42) TRPV1CYP1A2HSD11B1CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946559-A2 IMIDAZOPYRIDAZINES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1999-10-06 EP disclosed
WO-1998028299-A2 IMIDAZOPYRIDAZINES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-07-02 WO disclosed