SCHEMBL8089304

SCHEMBL8089304

Cc1cccnc1-n1ccnc1S

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
CYP2E1 P05181 1/20 0.39
CYP2A6 P11509 1/20 0.39
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
PSMD14 O00487 1/20 0.36
COPS5 Q92905 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HSD11B1 P28845 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8501020 0.81 CYP3A4 (0.53) CYP3A4CYP2E1CYP2A6NOS3NOS1
SCHEMBL8498987 0.79 RPS6KA5 (0.39) CYP3A4CYP2E1CYP2A6NOS3NOS1
SCHEMBL27536382 0.79 CYP3A4 (0.39) CYP3A4CYP2E1CYP2A6NOS3NOS1
SCHEMBL10685594 0.79 L3MBTL1 (0.36) CYP3A4CYP2E1CYP2A6KDM4ENPC1
SCHEMBL8699160 0.76 ALDH1A1 (0.42) CYP3A4CYP2E1CYP2A6L3MBTL1MAPT
SCHEMBL10723376 0.71 ADH5 (0.31)
SCHEMBL12369780 0.71 NOS3 (0.45) CYP2A6NOS3NOS1NOS2NPSR1
SCHEMBL10094619 0.70 CDC7 (0.50) NOS3NOS1NOS2NPSR1MEN1
SCHEMBL28661510 0.69 RPS6KA5 (0.47) NPSR1MEN1KMT2AMAPTRPS6KA5
SCHEMBL23196722 0.68 CYP3A4 (0.44) CYP3A4CYP2E1CYP2A6KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1105720-C Imidazopyridazines compound AOTANNA MEDICINE AG (DE) 2003-04-16 CN disclosed
US-6043242-A TREATING A MAMMAL AFFLICTED WITH A DISEASE BASED ON HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-03-28 US disclosed
CN-1246120-A Imidazopyridazines compound BYK GULDEN LOMBERG CHEM FAB (DE) 2000-03-01 CN disclosed
US-5053417-A Antiulcer agents TANABE SEIYAKU CO., LTD. (JP) 1991-10-01 US disclosed
US-4996217-A Antiulcer agents TANABE SEIYAKU COMPANY, LTD. (JP) 1991-02-26 US disclosed