SCHEMBL8501121

SCHEMBL8501121

CC(CC(=O)O)c1cccc(CNC(=O)c2cccc(NCC=[N+](N)C#N)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
FFAR1 O14842 1/20 0.38
ROCK2 O75116 4/20 0.38
GRK2 P25098 3/20 0.38
PRKCA P17252 2/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 2/20 0.37
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
ALOX5 P09917 1/20 0.36
EPHX2 P34913 1/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
HTT P42858 2/20 0.36
PPARG P37231 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856468 0.80 TP53 (0.46) TP53TSHRMEN1KMT2AFFAR1
SCHEMBL7864206 0.78 TP53 (0.45) TP53TSHRMEN1KMT2AFFAR1
SCHEMBL7856464 0.77 TP53 (0.49) TP53TSHRMEN1KMT2AROCK2
SCHEMBL7856412 0.75 TP53 (0.47) TP53TSHRMEN1KMT2AFFAR1
SCHEMBL7350700 0.72 RAB9A (0.47) TP53MEN1KMT2AMAPK1HSD17B10
SCHEMBL7864178 0.71 TP53 (0.43) TP53TSHRSIRT2LMNAMAPK1
SCHEMBL7863185 0.71 AKR1C3 (0.56) MEN1KMT2ALMNAALDH1A1GAA
SCHEMBL7861566 0.70 ROCK2 (0.41) TP53TSHRROCK2GRK2PRKCA
SCHEMBL7864712 0.69 SIRT2 (0.45) SIRT2LMNAMAPK1HSD17B10ALDH1A1
SCHEMBL7864751 0.69 SIRT2 (0.41) TP53TSHRSIRT2LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed