SCHEMBL7864751

SCHEMBL7864751

CCC(CC(=O)O)c1cccc(CNC(=O)c2cccc(NC=NN)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.41
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41
LMNA P02545 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CFD P00746 1/20 0.40
MAPK1 P28482 1/20 0.40
SENP1 Q9P0U3 4/20 0.40
SENP2 Q9HC62 1/20 0.40
PPARG P37231 1/20 0.40
POLB P06746 1/20 0.39
MMP13 P45452 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ITGB3 P05106 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856468 0.88 TP53 (0.46) SIRT2TP53TSHRLMNAALDH1A1
SCHEMBL7864712 0.87 SIRT2 (0.45) SIRT2LMNAALDH1A1GAAHSD17B10
SCHEMBL7864673 0.87 MAPT (0.42) LMNAGAAPPARGHTT
SCHEMBL7864178 0.86 TP53 (0.43) SIRT2TP53TSHRLMNAALDH1A1
SCHEMBL7862019 0.85 LMNA (0.45) SIRT2TP53TSHRLMNAALDH1A1
SCHEMBL7866898 0.85 ALDH1A1 (0.42) ALDH1A1GAAPPARGHTTHDAC8
SCHEMBL7864322 0.83 AURKA (0.41) SIRT2TP53TSHRLMNAALDH1A1
SCHEMBL7864771 0.82 MAPT (0.46) SIRT2TP53LMNAALDH1A1GAA
SCHEMBL7864776 0.82 PPARG (0.53) LMNAPPARG
SCHEMBL7856483 0.81 SIRT2 (0.48) SIRT2LMNAALDH1A1GAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed