SCHEMBL8501867

SCHEMBL8501867

CCOC(=O)[S+]([O-])CCOc1ccnc(C[S+]([O-])c2nc3ccccc3[nH]2)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
KMT2A Q03164 5/20 0.44
MAPT P10636 5/20 0.44
CYP2C9 P11712 4/20 0.44
LMNA P02545 4/20 0.44
WDR5 P61964 3/20 0.44
ENGASE Q8NFI3 3/20 0.44
HPGD P15428 3/20 0.44
DDAH1 O94760 2/20 0.44
ADORA3 P0DMS8 2/20 0.44
TBXA2R P21731 2/20 0.44
NPY1R P25929 2/20 0.44
ADORA1 P30542 2/20 0.44
OPRM1 P35372 2/20 0.44
HTR3A P46098 2/20 0.44
FASN P49327 2/20 0.44
SARM1 Q6SZW1 2/20 0.44
ABCG2 Q9UNQ0 2/20 0.44
HTR1A P08908 1/20 0.44
IDE P14735 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8500264 0.88 KMT2A (0.48) ALDH1A1KMT2AMAPTCYP2C9LMNA
SCHEMBL8526311 0.87 ALDH1A1 (0.43) ALDH1A1KMT2AMAPTCYP2C9LMNA
SCHEMBL8502342 0.86 KMT2A (0.46) ALDH1A1KMT2AMAPTCYP2C9LMNA
SCHEMBL9022527 0.86 KMT2A (0.48) ALDH1A1KMT2AMAPTCYP2C9LMNA
SCHEMBL13871335 0.86 CYP2C9 (0.46) ALDH1A1KMT2AMAPTCYP2C9LMNA
SCHEMBL6476745 0.85 KMT2A (0.46) ALDH1A1KMT2AMAPTCYP2C9LMNA
SCHEMBL8503283 0.85 LMNA (0.47) ALDH1A1KMT2AMAPTCYP2C9LMNA
SCHEMBL6582664 0.85 KMT2A (0.49) ALDH1A1KMT2AMAPTCYP2C9LMNA
SCHEMBL9025491 0.84 KMT2A (0.45) ALDH1A1KMT2AMAPTCYP2C9LMNA
SCHEMBL8542308 0.84 KMT2A (0.49) ALDH1A1KMT2AMAPTCYP2C9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998445-A PEPTIC ULCERS EISAI CO., LTD. (JP) 1999-12-07 US disclosed
US-5840910-A Pyridine derivatives having anti-ulcerative activity ESAI CO., LTD. (JP) 1998-11-24 US disclosed
EP-0654471-A1 Pyridine derivatives, pharmaceutical compositions comprising the same, the use of the same for the manufacture of medicaments having therapeutic or preventative value, and process for preparing the same Eisai Co., Ltd. (JP) 1995-05-24 EP disclosed
US-5045552-A Pyridine derivatives having anti-ulcerative activity EISAI CO., LTD. (JP) 1991-09-03 US disclosed