SCHEMBL8502147

SCHEMBL8502147

O=C(O)C(CCO)(CSc1ccc(O)cc1)c1ccc(-c2ccc(Cl)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
RET P07949 1/20 0.37
MAPT P10636 3/20 0.35
NPC1 O15118 2/20 0.35
GAA P10253 2/20 0.35
RAB9A P51151 2/20 0.35
MAPK1 P28482 2/20 0.35
KMT2A Q03164 1/20 0.35
MMP2 P08253 4/20 0.34
MMP3 P08254 3/20 0.34
MMP9 P14780 3/20 0.34
MMP13 P45452 2/20 0.34
MMP1 P03956 1/20 0.34
MMP8 P22894 1/20 0.34
CYP2C19 P33261 2/20 0.33
LMNA P02545 1/20 0.33
HSP90AA1 P07900 1/20 0.33
THRB P10828 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8505537 0.90 MMP2 (0.43) KDM4EALDH1A1MAPTNPC1RAB9A
SCHEMBL8502321 0.84 RET (0.39) KDM4EALDH1A1RETMAPTNPC1
SCHEMBL11215216 0.77 ESR1 (0.49) ALDH1A1MAPK1CYP2C19LMNACYP1A2
SCHEMBL8690818 0.74 MMP2 (0.42) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL7353635 0.74 MMP2 (0.42) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL7353628 0.74 MMP2 (0.42) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL8502365 0.70 CNR1 (0.40) ALDH1A1MAPTMIF
SCHEMBL8504171 0.67 MMP2 (0.57) ALDH1A1MAPTKMT2AMMP2MMP3
SCHEMBL7996868 0.64 KDM4E (0.51) KDM4EALDH1A1RETMAPTNPC1
SCHEMBL6784818 0.63 ESR1 (0.42) ALDH1A1MAPTNPC1GAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939583-A ANTIARTHRITIC AGENTS; BONE, CARDIOVASCULAR, BRAIN, NERVOUS SYSTEM DISORDERS; ANTITUMOR AND ANTIMETASTASIS AGENTS BAYER CORPORATION (US) 1999-08-17 US claimed
US-5939583-A ANTIARTHRITIC AGENTS; BONE, CARDIOVASCULAR, BRAIN, NERVOUS SYSTEM DISORDERS; ANTITUMOR AND ANTIMETASTASIS AGENTS BAYER CORPORATION (US) 1999-08-17 US disclosed