SCHEMBL8503418

SCHEMBL8503418

N=C(N)c1ccc(C(N)(CCC=O)C(=O)O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.45
CYP1A2 P05177 1/20 0.45
KMT2A Q03164 1/20 0.45
F2 P00734 3/20 0.40
PRSS1 P07477 3/20 0.40
PRSS2 P07478 3/20 0.40
PRSS3 P35030 3/20 0.40
PLG P00747 1/20 0.40
C1S P09871 1/20 0.40
NQO2 P16083 2/20 0.38
CPN1 P15169 1/20 0.37
CPB2 Q96IY4 1/20 0.37
PRMT5 O14744 1/20 0.36
PRMT1 Q99873 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GRM5 P41594 1/20 0.36
GRM1 Q13255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8497829 0.99 KMT2A (0.44) MEN1CYP1A2KMT2AF2PRSS1
SCHEMBL8905131 0.85 MEN1 (0.47) MEN1CYP1A2KMT2AF2PRSS1
Hydrochloric Acid SCHEMBL8500969 0.84 KMT2A (0.46) MEN1CYP1A2KMT2AF2PRSS1
SCHEMBL6011852 0.78 MEN1 (0.73) MEN1CYP1A2KMT2AF2PRSS1
SCHEMBL8503420 0.75 MEN1 (0.38) MEN1CYP1A2KMT2AGRM5GRM1
Hydrochloric Acid SCHEMBL8497837 0.74 MEN1 (0.37) MEN1CYP1A2KMT2A
SCHEMBL27403702 0.69 F2 (0.47) F2PRSS1PRSS2PRSS3PLG
SCHEMBL10604183 0.69 NQO2 (0.51) MEN1CYP1A2KMT2AF2PRSS1
SCHEMBL1445807 0.67 PRSS1 (0.53) F2PRSS1PRSS2PRSS3PLG
SCHEMBL8501113 0.67 PRMT5 (0.38) F2PRSS1PRSS2PRSS3PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5886208-A Substituted B-amino acid derivatives useful as platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1999-03-23 US disclosed
US-5703125-A MELT BLEND OF SOAP, SURFACTANT AND SOLVENT G. D. SEARLE & CO. (US) 1997-12-30 US disclosed