SCHEMBL850992

SCHEMBL850992

C[C@H](N)[C@H](O)Cc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.63
SLC6A2 P23975 2/20 0.61
TAAR1 Q96RJ0 2/20 0.61
MAOA P21397 1/20 0.61
SLC6A4 P31645 1/20 0.61
SLC6A3 Q01959 1/20 0.61
SIGMAR1 Q99720 1/20 0.61
CYP2A6 P11509 1/20 0.61
ADORA2A P29274 1/20 0.61
ADORA1 P30542 1/20 0.61
TRPA1 O75762 2/20 0.57
EPHX1 P07099 1/20 0.54
CSNK1E P49674 1/20 0.50
ALPI P09923 1/20 0.50
PKM P14618 1/20 0.50
PTGS1 P23219 1/20 0.50
XIAP P98170 1/20 0.50
SLC7A5 Q01650 1/20 0.50
ADRA2A P08913 1/20 0.48
ADRA2C P18825 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9816875 1.00 CYP2D6 (0.63) CYP2D6SLC6A2TAAR1MAOASLC6A4
SCHEMBL20179498 1.00 CYP2D6 (0.63) CYP2D6SLC6A2TAAR1MAOASLC6A4
Hydrochloric Acid SCHEMBL835498 0.98 CYP2D6 (0.61) CYP2D6SLC6A2TAAR1MAOASLC6A4
SCHEMBL15640342 0.83 SLC6A2 (0.57) CYP2D6SLC6A2TAAR1MAOASLC6A4
SCHEMBL1168783 0.83 SLC6A2 (0.57) CYP2D6SLC6A2TAAR1MAOASLC6A4
SCHEMBL11163544 0.82 EPHX1 (0.58) CYP2D6SLC6A2TAAR1MAOASLC6A4
SCHEMBL873142 0.82 TRPA1 (0.61) CYP2D6SLC6A2TAAR1MAOASLC6A4
SCHEMBL107335 0.82 TRPA1 (0.61) CYP2D6SLC6A2TAAR1MAOASLC6A4
SCHEMBL26085425 0.82 TRPA1 (0.61) CYP2D6SLC6A2TAAR1MAOASLC6A4
SCHEMBL26085426 0.82 TRPA1 (0.61) CYP2D6SLC6A2TAAR1MAOASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120252770-A1 Chemical Compounds 572 BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-10-04 US disclosed
US-20120252770-A1 Chemical Compounds 572 BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-10-04 US disclosed
US-8143290-B2 Chemical compounds 572 ASTRAZENECA AB (SE) 2012-03-27 US disclosed
US-20110071194-A1 Chemical Compounds 572 BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-03-24 US disclosed
US-20100197644-A1 Chemical Compounds 572 BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2010-08-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197644-A1 Chemical Compounds 572 ABCG2, ABCB1, CYP11B2 CYP2D6 17/4885SLC6A2 3062/4885TAAR1 4379/4885
US-20120252770-A1 Chemical Compounds 572 ABCG2, ABCB1, CYP11B2 CYP2D6 17/4885SLC6A2 3062/4885TAAR1 4379/4885
US-20110071194-A1 Chemical Compounds 572 ABCG2, ABCB1, CYP11B2 CYP2D6 17/4885SLC6A2 3062/4885TAAR1 4379/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.