SCHEMBL851003

SCHEMBL851003

N#Cc1cccc(Oc2ccccc2C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.51
CCR2 P41597 1/20 0.49
ALDH1A1 P00352 1/20 0.49
KDM4E B2RXH2 1/20 0.48
POLB P06746 1/20 0.48
CTNNB1 P35222 1/20 0.47
PYGL P06737 1/20 0.47
PYGM P11217 1/20 0.47
XDH P47989 1/20 0.47
SLC22A12 Q96S37 1/20 0.47
AKR1C3 P42330 1/20 0.45
F7 P08709 1/20 0.44
F3 P13726 1/20 0.44
EPAS1 Q99814 2/20 0.43
NOTUM Q6P988 1/20 0.43
STK10 O94804 1/20 0.43
SLK Q9H2G2 1/20 0.43
MGLL Q99685 1/20 0.43
VEGFA P15692 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30728621 0.87 HTT (0.45) HTTKDM4EPOLBPYGLPYGM
SCHEMBL7695689 0.87 CTNNB1 (0.62) ALDH1A1KDM4ECTNNB1EPAS1VEGFA
SCHEMBL28949714 0.87 CTNNB1 (0.43) HTTCTNNB1PYGLPYGMEPAS1
SCHEMBL28949718 0.85 ALDH1A1 (0.43) HTTALDH1A1CTNNB1PYGLPYGM
SCHEMBL18772927 0.85 AR (0.45) HTTALDH1A1KDM4EPOLBEPAS1
SCHEMBL28560551 0.84 KDM4E (0.63) HTTALDH1A1KDM4EPOLBCTNNB1
SCHEMBL28011402 0.83 XDH (0.46) HTTKDM4EPOLBPYGLPYGM
SCHEMBL851138 0.83 CTNNB1 (0.51) HTTCCR2ALDH1A1KDM4EPOLB
SCHEMBL28264707 0.82 KDM4E (0.61) HTTALDH1A1KDM4EPOLBCTNNB1
SCHEMBL8432193 0.82 AR (0.55) SLC22A12EPAS1STK10SLKVEGFA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432556-A1 PROTEASE INHIBITORS Orion Corporation (FI) 2012-03-28 EP disclosed
WO-2010133748-A1 PROTEASE INHIBITORS ORION CORPORATION (FI) 2010-11-25 WO disclosed