SCHEMBL8511573

SCHEMBL8511573

Cc1c(-c2ccc(-c3ccc(OC(F)(F)F)cc3)nc2)nc2ccccc2c1OC(=O)N1CCOCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
KMT2A Q03164 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 3/20 0.41
TSHR P16473 2/20 0.41
USP2 O75604 2/20 0.41
TP53 P04637 2/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
POLB P06746 1/20 0.41
TRPV1 Q8NER1 1/20 0.40
EPHX1 P07099 1/20 0.40
CASP3 P42574 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
PPARD Q03181 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8515384 0.79 ACP1 (0.44) TRPV1ACP1SCN2ASCN10A
SCHEMBL8515625 0.78 ACP1 (0.45) TRPV1ADORA2AACP1SCN2ASCN10A
SCHEMBL8515434 0.76 HSD17B10 (0.43) KDM4ETSHRHSD17B10POLBMCHR1
SCHEMBL8514932 0.73 DHODH (0.49) TSHRACP1
SCHEMBL8514929 0.73 DHODH (0.49) TSHRACP1
SCHEMBL9607436 0.73 ACP1 (0.40) PPARDACP1CTNNB1SCN2ASCN10A
SCHEMBL8514251 0.71 PDE10A (0.44) TSHRPPARDPPARAACP1CTNNB1
SCHEMBL8514255 0.71 PDE10A (0.44) TSHRPPARDPPARAACP1CTNNB1
SCHEMBL8512120 0.68 SCN9A (0.45) ACP1CTNNB1
SCHEMBL28253958 0.68 PDE10A (0.48) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed