SCHEMBL8512658

SCHEMBL8512658

CC1(C)CCC(C)(C)c2cc(-c3ccnc(-c4ccncc4)c3)ccc21

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RARA P10276 13/20 0.44
RARB P10826 12/20 0.44
RARG P13631 11/20 0.43
RXRA P19793 3/20 0.42
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
NPC1 O15118 1/20 0.38
MAPKAPK2 P49137 1/20 0.37
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18961191 0.92 RARA (0.47) RARARARBRARGRXRAABCB1
SCHEMBL16998862 0.85 RARB (0.55) RARARARBRARGRXRAABCB1
SCHEMBL8510939 0.84 RARA (0.42) RARARARBRARGRXRAABCB1
SCHEMBL8513591 0.82 RARA (0.38) RARARARBRARGRXRAABCB1
Hydrochloric Acid SCHEMBL8510905 0.81 RARA (0.38) RARARARBRARGRXRAABCB1
SCHEMBL8514253 0.81 NPC1 (0.55) RARARARBRARGRXRAABCB1
SCHEMBL16998655 0.80 RARB (0.49) RARARARBRARGRXRAABCB1
SCHEMBL16998453 0.79 CCR1 (0.50) RARARARBRARGRXRAABCB1
SCHEMBL2015591 0.79 RARA (0.44) RARARARBRARGRXRAABCB1
SCHEMBL25791320 0.79 RARA (0.48) RARARARBRARGRXRAABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed