SCHEMBL8514253

SCHEMBL8514253

CC1(C)CCC(C)(C)c2cc(-c3ccnc(-c4ccncc4)n3)ccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.55
RARB P10826 8/20 0.50
RARA P10276 8/20 0.50
RARG P13631 8/20 0.44
GABRA1 P14867 1/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
GABRA5 P31644 1/20 0.43
GABRA3 P34903 1/20 0.43
KMT2A Q03164 5/20 0.41
MEN1 O00255 4/20 0.41
MAPT P10636 3/20 0.41
POLB P06746 3/20 0.41
KDM4E B2RXH2 2/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RXRA P19793 3/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8511483 0.84 RARB (0.46) NPC1RARBRARARARGKMT2A
SCHEMBL8512804 0.84 RARA (0.49) NPC1RARBRARARARGKMT2A
SCHEMBL8515301 0.84 NPC1 (0.40) NPC1RARBRARA
SCHEMBL8515254 0.83 RARB (0.51) NPC1RARBRARARARGKMT2A
SCHEMBL31060783 0.83 RARB (0.51) NPC1RARBRARARARGKMT2A
SCHEMBL9612772 0.82 RARB (0.47) NPC1RARBRARARARGKMT2A
SCHEMBL8511696 0.82 RARB (0.44) NPC1RARBRARARARGKMT2A
Hydrochloric Acid SCHEMBL8515237 0.81 RARB (0.44) NPC1RARBRARARARGKMT2A
SCHEMBL8512658 0.81 RARA (0.44) NPC1RARBRARARARGRXRA
SCHEMBL8510213 0.81 RARA (0.50) RARBRARARARGPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed