SCHEMBL8512705

SCHEMBL8512705

Cc1nn(-c2cccc(N)c2)c(C)c1CC(=O)O

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
PTGDR2 Q9Y5Y4 1/20 0.54
P2RX7 Q99572 17/20 0.52
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3828501 0.86 NPC1 (0.57) NPC1RAB9APTGDR2P2RX7TSHR
SCHEMBL11253889 0.85 P2RX7 (0.59) NPC1RAB9APTGDR2P2RX7
SCHEMBL1195590 0.84 NPC1 (0.73) NPC1RAB9APTGDR2P2RX7TSHR
SCHEMBL9609107 0.83 P2RX7 (0.47) NPC1RAB9APTGDR2P2RX7TSHR
SCHEMBL11250187 0.81 P2RX7 (0.57) NPC1RAB9APTGDR2P2RX7
SCHEMBL8511047 0.80 PDE4B (0.62) NPC1RAB9APTGDR2P2RX7
SCHEMBL11539322 0.77 RAB9A (0.58) NPC1RAB9APTGDR2P2RX7TSHR
SCHEMBL1195287 0.77 P2RX7 (0.57) NPC1RAB9APTGDR2P2RX7TSHR
SCHEMBL8514171 0.77 PTGDR2 (0.62) PTGDR2
SCHEMBL8512906 0.77 NPC1 (0.62) NPC1RAB9APTGDR2P2RX7TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069175-A1 NEW PYRAZOLE DERIVATIVES HAVING CRTH2 ANTAGONISTIC BEHAVIOUR ALMIRALL, S.A. (ES) 2012-05-31 WO disclosed