SCHEMBL8512706

SCHEMBL8512706

Cc1ccc(F)cc1S(=O)(=O)N1CCN(C(=O)O)CC1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.54
RAB9A P51151 1/20 0.54
NOD1 Q9Y239 1/20 0.54
SMN1; SMN2 Q16637 5/20 0.53
TDP1 Q9NUW8 1/20 0.52
MAPT P10636 3/20 0.51
TP53 P04637 3/20 0.51
MAPK1 P28482 2/20 0.51
HTT P42858 1/20 0.51
ALDH1A1 P00352 2/20 0.51
CNR2 P34972 1/20 0.50
POLB P06746 1/20 0.50
ATM Q13315 1/20 0.50
PKM P14618 2/20 0.49
TSHR P16473 1/20 0.49
CNR1 P21554 1/20 0.48
KDM4E B2RXH2 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2081383 0.85 TNF (0.51) TNFRAB9ANOD1SMN1; SMN2TDP1
SCHEMBL4166290 0.81 ALDH1A1 (0.67) TNFRAB9ANOD1SMN1; SMN2MAPT
SCHEMBL11888841 0.80 SMN1; SMN2 (0.51) TNFRAB9ANOD1SMN1; SMN2MAPT
SCHEMBL8516111 0.80 ALDH1A1 (0.46) SMN1; SMN2ALDH1A1POLBPKMTSHR
SCHEMBL2080681 0.78 TP53 (0.65) SMN1; SMN2MAPTTP53ALDH1A1CNR2
SCHEMBL2081742 0.78 ALDH1A1 (0.73) SMN1; SMN2MAPTTP53MAPK1HTT
SCHEMBL5246389 0.75 MAPT (0.66) SMN1; SMN2MAPTTP53POLBTSHR
SCHEMBL29060784 0.74 PKM (0.66) SMN1; SMN2TDP1MAPK1ALDH1A1POLB
SCHEMBL18711646 0.73 ALDH1A1 (0.76) RAB9AMAPTMAPK1ALDH1A1PKM
SCHEMBL2079086 0.73 NPC1 (0.76) RAB9ASMN1; SMN2MAPTTP53HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069175-A1 NEW PYRAZOLE DERIVATIVES HAVING CRTH2 ANTAGONISTIC BEHAVIOUR ALMIRALL, S.A. (ES) 2012-05-31 WO disclosed
EP-2457900-A1 New pyrazole derivatives having CRTh2 antagonistic behaviour Almirall, S.A. (ES) 2012-05-30 EP disclosed